Gisadenafil besylate

Catalog # Availability Size / Price Qty
4165/10
4165/50
Gisadenafil besylate | CAS No. 334827-98-4 | Phosphodiesterase Inhibitors
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Description: Potent PDE5 inhibitor; orally bioavailable
Alternative Names: UK 369003

Chemical Name: 5-[2-Ethoxy-5-[(4-ethyl-1-piperazinyl)sulfonyl]-3-pyridinyl]-3-ethyl-2,6-dihydro-2-(2-methoxyethyl)-7H-pyrazolo[4,3-d]pyrimidin-7-one benzenesulfonate

Purity: ≥99%

Product Details
Citations (1)
Reviews

Biological Activity

Potent PDE5 inhibitor (IC50 = 1.23 nM). Shows >100-fold selectivity for PDE5 over PDE6. Orally bioavailable.

Technical Data

M.Wt:
677.79
Formula:
C23H33N7O5S.C6H6O3S
Solubility:
Soluble to 10 mM in water and to 100 mM in DMSO
Purity:
≥99%
Storage:
Desiccate at RT
CAS No:
334827-98-4

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.

Additional Information

Licensing Caveats:
Sold for research purposes under agreement from Pfizer Inc.

Product Datasheets

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Citation for Gisadenafil besylate

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