receptor agonist; Ki
values are 7.6 and 900 nM for CB2
receptors respectively. Increases P-ERK1/2 expression in HL-60 cells in vitro
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Tricyclic pyrazoles. 4. Synthesis and biological evaluation of analogues of the robust and selective CB2 cannabinoid ligand 1-(2',4'-dichlorophenyl)-6-methyl-N-piperidin-1-yl-1,4-dihydroindeno[1,2-c]pyrazole-3-carboxam
Murineddu et al.