Chemical Name: N-[2-Methyl-5-(1-piperidinylsulfonyl)-3-furanyl]-N'-phenylurea
Biological ActivityGSK 264220A is an endothelial lipase and lipoprotein lipase inhibitor (IC50 values are 0.13 and 0.10 μM respectively).
The technical data provided above is for guidance only.
For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.
A high-throughput screen for the endothelial lipase using HDL as substrate.
Keller et al.
Discovery of potent, selective sulfonylfuran urea endothelial lipase inhibitors.
Goodman et al.
Citation for GSK 264220A
The citations listed below are publications that use Tocris products. Selected citations for GSK 264220A include:
1 Citation: Showing 1 - 1
Analysis of ECs and related compounds in plasma: artifactual isomerization and ex vivo enzymatic generation of 2-MGs.
Authors: Pastor Et al.
J Lipid Res 2014;55:966
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