GSK 264220A

Catalog # Availability Size / Price Qty
GSK 264220A | CAS No. 685506-42-7 | Lipase Inhibitors
1 Image
Description: Endothelial lipase and lipoprotein lipase inhibitor

Chemical Name: N-[2-Methyl-5-(1-piperidinylsulfonyl)-3-furanyl]-N'-phenylurea

Purity: ≥98%

Product Details
Citations (1)

Biological Activity

GSK 264220A is an endothelial lipase and lipoprotein lipase inhibitor (IC50 values are 0.13 and 0.10 μM respectively).

Technical Data

Soluble to 100 mM in DMSO and to 10 mM in ethanol
Store at +4°C

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.

Background References

  1. A high-throughput screen for the endothelial lipase using HDL as substrate.
    Keller et al.
    J.Biomol.Screen., 2008;13:468
  2. Discovery of potent, selective sulfonylfuran urea endothelial lipase inhibitors.
    Goodman et al.
    Bioorg.Med.Chem.Letts., 2009;19:27

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Citation for GSK 264220A

The citations listed below are publications that use Tocris products. Selected citations for GSK 264220A include:

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