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GSK 3787

Catalog #: 3961
1 Citation Datasheet / COA / SDS
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3961/50
GSK 3787 | CAS No. 188591-46-0 | PPAR delta Receptor Antagonists
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Description: Potent and selective PPARδ antagonist

Chemical Name: 4-Chloro-N-[2-[[5-(trifluoromethyl)-2-pyridinyl]sulfonyl]ethyl]benzamide

Purity: ≥99%

Product Details
Citations (1)
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Biological Activity

GSK 3787 is a potent and selective peroxisome proliferator-activated receptor δ (PPARδ) antagonist (pIC50 = 6.6). Displays no measurable affinity for PPARα or PPARγ in vitro (pIC50< 5).

Technical Data

M.Wt:
392.78
Formula:
C15H12ClF3N2O3S
Solubility:
Soluble to 100 mM in DMSO
Purity:
≥99%
Storage:
Store at +4°C
CAS No:
188591-46-0

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.

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Citation for GSK 3787

The citations listed below are publications that use Tocris products. Selected citations for GSK 3787 include:

1 Citation: Showing 1 - 1

  1. PPARδ signaling mediates the cytotoxicity of DHA in H9c2 cells.
    Authors: Samokhvalov Et al.
    Cell Cycle  2015;232:44105

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VersaClone cDNA Plasmids

Human PPAR delta/NR1C2 (NP_006229) VersaClone cDNA

RDC2078

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