Very selective β2
adrenergic antagonist (Ki
values are 1.2, 120 and 257 nM for β2
receptors respectively). Active in vivo
. Also available as part of the β-Adrenoceptor Antagonist Tocriset™
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
All Tocris products are intended for laboratory research use only.
Sold with the permission of AstraZeneca UK Ltd.
Function and regulation of the β3-adrenoceptor.
Strosberg and Pietri-Rouxel
The pharmacology of a β2-selective adrenoceptor antagonist (ICI-118,551).
Bilski et al.
β-Adrenoceptor subtypes and the opening of plasmalemmal K+-channels in trachealis muscle: electrophysiological and mechanical studies in guinea-pig tissue.
Cook et al.
β2-but not β3-adrenoceptors mediate prejunctional inhibition of non-adrenergic non cholinergic contraction of guinea pig main bronchi.
Ten Berge et al.
The citations listed below are publications that use Tocris products. Selected citations for ICI 118,551 hydrochloride include:
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