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Idazoxan hydrochloride

Catalog #: 0793
2 Citations Datasheet / COA / SDS

Discontinued Product

0793 has been discontinued.
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Idazoxan hydrochloride | CAS No. 79944-56-2 | Adrenergic alpha-2 Receptor Antagonists
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Description: α2 antagonist. Also I2 ligand
Alternative Names: RX 781094

Chemical Name: 2-(1,4-Benzodioxan-2-yl)-2-imidazoline hydrochloride

Purity: ≥98%

Product Details
Citations (2)
Reviews
Biological Activity Technical Data Background Product Datasheets Calculators

Biological Activity

Idazoxan hydrochloride is a α2-adrenoceptor antagonist, and I2 ligand, selective over I1 sites (pKi values are 5.90, 7.22, 8.01, 7.43, and 7.7 for I1, I2, α2A, α2B, and α2C receptors respectively).

Technical Data

M.Wt:
240.69
Formula:
C11H12N2O2.HCl
Solubility:
Soluble to 100 mM in water
Purity:
≥98%
Storage:
Store at RT
CAS No:
79944-56-2

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.

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Product Datasheets

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Citations for Idazoxan hydrochloride

The citations listed below are publications that use Tocris products. Selected citations for Idazoxan hydrochloride include:

2 Citations: Showing 1 - 2

  1. μ-Opioid receptor activation and noradrenaline transport inhibition by tapen. in rat single locus coeruleus neurons.
    Authors: Sadeghi Et al.
    Development  2015;172:460
  2. Medullary NE neurons modulate local oxygen concentrations in the bed nucleus of the stria terminalis.
    Authors: Bucher Et al.
    J Cereb Blood Flow Metab  2014;34:1128

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