A moderately potent, but highly selective α2
-adrenoceptor antagonist, the only reported selective antagonist at the α2B
-adrenoceptor not having potent α1
-adrenoceptor antagonist activity.
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Assessment of imiloxan as a selective α2B-adrenoceptor antagonist.
Michel et al.
2-(2-Imidazolylmethyl)-1,4-benzodioxans, a series of selective alpha2-adrenoceptor antagonists.
Michel and Whiting