Imiloxan hydrochloride

Key Product Details

Product Description

Imiloxan hydrochloride is a moderately potent, but highly selective α₂-adrenoceptor antagonist, the only reported selective antagonist at the α_2B-adrenoceptor not having potent α₁-adrenoceptor antagonist activity.

Licensing Information

Sold with the permission of Roche Bioscience

Product Specifications for Imiloxan hydrochloride

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.

Solubility

Preparing Stock Solutions for Imiloxan hydrochloride

The following data is based on the product molecular weight 280.75.

Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which all affect the solvent volumes required to prepare stock solutions.

Select a batch to recalculate based on the batch molecular weight:

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Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
1 mM	3.56 mL	17.81 mL	35.62 mL
5 mM	0.71 mL	3.56 mL	7.12 mL
10 mM	0.36 mL	1.78 mL	3.56 mL
50 mM	0.07 mL	0.36 mL	0.71 mL

Calculators

Background References

References are publications that support the biological activity of the product. See our Citations tab to view 5 publications citing the usage of this product.

• Michel and Whiting 2-(2-Imidazolylmethyl)-1,4-benzodioxans, a series of selective alpha₂-adrenoceptor antagonists. Br.J.Pharmacol.
• Michel Assessment of imiloxan as a selective α_2B-adrenoceptor antagonist. Br.J.Pharmacol. 1990 PMID: 1970500

Product Documents for Imiloxan hydrochloride