Catalog Number: 0992
Chemical Name: 1-[(1-Methylethyl)amino]-3-[2-(1H-pyrrol-1-yl)]-propan-2-ol hemifumarate
Biological Activity
5-HT1B antagonist, approximately 30-fold selective over 5-HT1A. Also possesses affinity for β-adrenergic receptors.
Technical Data
  • M.Wt:
    332.4
  • Formula:
    C16H22N2O2.½C4H4O4
  • Solubility:
    Soluble to 10 mM in water with gentle warming
  • Purity:
    >99%
  • Storage:
    Desiccate at +4°C
  • CAS No:
    874882-92-5
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis. All Tocris products are intended for laboratory research use only.
Background References
  1. Interactions of isamoltane (CGP 361A), an anxiolytic phenoxypropanolamine derivative, with 5-HT1 receptor subtypes in the rat brain.
    Waldmeier et al.
    Naunyn Schmiedebergs Arch.Pharmacol., 1988;337:609

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