5-HT1B Receptor Antagonists: Products

5-HT1B is a 7TM receptor for serotonin and is expressed on striatal neurons and Purkinje cells in the cerebellum. 5-HT1B ligation inhibits glycinergic signaling, appetite, circadian rhythym light responsiveness, and trigeminal-mediated nociception.

"5-HT1B Receptor Antagonists" has 10 results in Products.
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SB 224289 hydrochloride 

Selective 5-HT1B antagonist


Selective r5-HT1B antagonist; active in vivo

GR 127935 hydrochloride 

Potent and selective 5-HT1B and 5-HT1D antagonist

Isamoltane hemifumarate 

5-HT1B antagonist

Cyanopindolol hemifumarate 

5-HT1A and 5-HT1B antagonist; also β-adrenergic antagonist

GR 55562 dihydrochloride 

5-HT1B antagonist


β3 partial agonist; also 5-HT1A and 5-HT1B antagonist; more active enantiomer of pindolol (Cat. No. 0994)

SB 216641 hydrochloride 

Selective h5-HT1B antagonist

SDZ 21009 

β-adrenoceptor antagonist; also 5-HT1A and 5-HT1B antagonist

LY 393558 

Dual 5-HT1B and 5-HT1D antagonist; also 5-HT re-uptake inhibitor
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