Biological Activity[Leu5]-Enkephalin is an endogenous opioid agonist peptide; inhibits electrically stimulated contractions in mouse vas deferens (IC50 = 11.4 nM). Short-acting in vivo.
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Tocris products are intended for laboratory research use only, unless stated otherwise.
Synthesis and pharmacological characterization in vitro of cyclic enkephalin analogues: effect of conformational constraints on opiate receptor selectivity.
DiMaio et al.
Binding of Leu5-enkephalin and Met5-enkephalin to a particulate fraction from rat cerebrum.
Meunier et al.
FEBS Lett., 1977;77:209
3H-Leu5-enkephalin specific binding to synaptic membrane - comparison with 3H-dihydromorphine and 3H-naloxone.
Law and Loh
Citation for [Leu5]-Enkephalin
The citations listed below are publications that use Tocris products. Selected citations for [Leu5]-Enkephalin include:
1 Citation: Showing 1 - 1
N-glycan-mediated quality control in the endoplasmic reticulum is required for the expression of correctly folded delta-opioid receptors at the cell surface.
Authors: Markkanen and Petäjä-Repo
J Biol Chem 2008;283:29086
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