LY 2119620

Catalog # Availability Size / Price Qty
6964/50
6964/10
LY 2119620 | CAS No. 886047-22-9 | mAChR M4 Modulators
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Description: Positive allosteric modulator of M2 and M4 receptors

Chemical Name: 3-Amino-5-chloro-N-cyclopropyl-4-methyl-6-[2-(4-methyl-1-piperazinyl)-2-oxoethoxy]-thieno[2,3-b]pyridine-2-carboxamide

Purity: ≥98%

Product Details
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Biological Activity

Positive allosteric modulator of M2 and M4 muscarinic receptors. Potentiates activity of agonist at receptor in G protein-coupled functional assay. Cooperativity factor, α = 19.5 and 79.4 for M2 and M4 in presence of ACh, respectively. Binds in extracellular site.

Technical Data

M.Wt:
437.94
Formula:
C19H24ClN5O3S
Solubility:
Soluble to 100 mM in DMSO and to 100 mM in 1eq. HCl
Purity:
≥98%
Storage:
Store at -20°C
CAS No:
886047-22-9

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.

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