LY 225910

  ( 3 citations )    
Product Datasheet
Catalog Number:1018
Chemical Name:2-[2-(5-Bromo-1H-indol-3-yl)ethyl]-3-[3-(1-methylethoxy)phenyl]-4-(3H)-quinazoline
Product Details
Citations (3)
Supplemental Products
Reviews
Biological Activity
Potent CCK2 receptor antagonist (IC50 = 9.3 nM for inhibition of 125I-labeled CCK-8 sulfate binding at mouse brain membranes).
Technical Data
  • M.Wt:
    502.41
  • Formula:
    C27H24BrN3O2
  • Solubility:
    Soluble to 100 mM in DMSO
  • Storage:
    Desiccate at -20°C
  • CAS No:
    133040-77-4
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis. All Tocris products are intended for laboratory research use only.
Additional Information
Licensing Caveats:
Sold with the permission of Eli Lilly and Company.
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Citations:

The citations listed below are publications that use Tocris products. Selected citations for LY 225910 include:

3 Citations: Showing 1 - 3
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  1. Phencyclidine-induced social withdrawal results from deficient stimulation of cannabinoid CB1 receptors: implications for schizophrenia.
    Authors: Seillier Et al.
    Neuropharmacology  2013;38:1816
  2. Cholecystokinin inhibits endocannabinoid-sensitive hippocampal IPSPs and stimulates others.
    Authors: Karson Et al.
    J Card Fail  2008;54:117
  3. Cortical sources of CRF, NKB, and CCK and their effects on pyramidal cells in the neocortex.
    Authors: Gallopin Et al.
    Neuropsychopharmacology  2006;16:1440

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