Catalog Number: 2697
Alternate Names: Galanin(1-13)-Gln14-bradykinin(2-9)amide
Biological Activity
Selective galanin GAL1 receptor agonist (Ki values are 0.23 and 5.71 nM for GAL1 and GAL2 receptors respectively). Enhances food consumption in rats following i.c.v. administration and reduces CAP-induced inflammatory pain.
Technical Data
  • M.Wt:
    2361.68
  • Formula:
    C112H161N29O28
  • Sequence:
    GWTLNSAGYLLGPQPPGFSPFR

    (Modifications: Arg-22 = C-terminal amide)

  • Solubility:
    Soluble to 1 mg/ml in water
  • Storage:
    Store at -20°C
  • CAS No:
    860790-38-1
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis. All Tocris products are intended for laboratory research use only.
Background References
  1. Regulation of kindling epileptogenesis by hippocampal galanin type 1 and type 2 receptors: the effects of subtype-selective agonists and the role of G-protein-mediated signaling.
    Mazarati et al.
    J.Pharmacol.Exp.Ther., 2006;318:700
  2. Activation of peripheral galanin receptors: differential effects on nociception.
    Jimenez-Andrade et al.
    Pharmacol.Biochem.Behav., 2006;85:273
  3. A galanin receptor subtype 1 specific agonist.
    Lundstrom et al.
    Int.J.Pept.Res.Ther., 2005;11:17

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