Selective liver receptor homolog 1 (LRH1, NR5A2) inverse agonist (IC50
= 320 nM and maximum efficacy of 64% repression). Exhibits >31-fold selectivity over SF1.
Soluble to 50 mM in DMSO
Store at +4°C
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All Tocris products are intended for laboratory research use only.
Discovery of inverse agonists for the liver receptor homologue-1 (LRH1; NR5A2).
Busby et al.
Probe Reports from the NIH Molecular Libraries Program, 2010;