Selective adenosine A2B
receptor antagonist (Ki
values are 1.97, 16.8, 403, 503, 570 and 612 nM for hA2B
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
All Tocris products are intended for laboratory research use only.
Sold with the permission of the University of Virginia Patent Foundation
Anilide derivatives of an 8-phenylxanthine carboxylic congener are highly potent and selective antagonists at human A2B adenosine receptors.
Kim et al.
[3H]MRS 1754, a selective antagonist radioligand for A2B adenosine receptors.
Ji et al.
Adenosine receptor activation ameliorates type I diabetes.
Nemeth et al.
FASEB J., 2007;21:2380
The citations listed below are publications that use Tocris products. Selected citations for MRS 1754 include:
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