NVP CXCR2 20

Tocris Bioscience | Catalog # 5660

Potent and selective CXCR2 antagonist
Tocris Bioscience
Discontinued Product
5660 has been discontinued. View all Chemokine Receptor Antagonists products.

Key Product Details

Description

Potent and selective CXCR2 antagonist

Product Description

Potent and selective CXCR2 antagonist (IC50 = 40 nM). Exhibits selectivity for CXCR2 over a panel of 49 other GPCRs. Orally bioavailable.

Product Specifications for NVP CXCR2 20

Molecular Weight

319.33

Formula

C15H11F2N3OS

Storage

Store at +4°C

Purity

≥98% (HPLC)

Chemical Name

4-Cyclopropyl-2-[[(2,3-difluorophenyl)methyl]thio]-1,6-dihydro-6-oxo5-pyrimidinecarbonitrile

CAS Number

1029521-30-9

PubChem ID

24955240

InChI Key

PHHZYKZFEBRXAL-UHFFFAOYSA-N

SMILES

OC1=C(C#N)C(C2CC2)=NC(SCC3=CC=CC(F)=C3F)=N1

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.

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Solubility

Solvent Max Conc. mg/mL Max Conc. mM
Solubility
DMSO 15.97 50

Preparing Stock Solutions for NVP CXCR2 20

The following data is based on the product molecular weight 319.33.

Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which all affect the solvent volumes required to prepare stock solutions.

Select a batch to recalculate based on the batch molecular weight:

Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.5 mM 6.26 mL 31.32 mL 62.63 mL
2.5 mM 1.25 mL 6.26 mL 12.53 mL
5 mM 0.63 mL 3.13 mL 6.26 mL
25 mM 0.13 mL 0.63 mL 1.25 mL

Calculators

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Background References

References are publications that support the biological activity of the product.

Product Documents for NVP CXCR2 20

Certificate of Analysis

To download a Certificate of Analysis, please enter a lot or batch number in the search box below.

Product Specific Notices for NVP CXCR2 20

For research use only

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