PD 102807

Tocris Bioscience | Catalog # 1671

Selective M4 antagonist
Tocris Bioscience

Key Product Details

Description

Selective M4 antagonist
View all mAChR M4 Antagonists »

Product Description

PD 102807 is a selective M4 muscarinic receptor antagonist. IC50 values are 91, 6559, 3441, 950 and 7412 nM for human M4, M1, M2, M3, and M5 receptors respectively. Promotes self-renewal of erythroid progenitors.

Product Specifications for PD 102807

Molecular Weight

392.45

Formula

C23H24N2O4

Storage

Store at RT

Purity

≥98% (HPLC)

Chemical Name

3,6a,11,14-Tetrahydro-9-methoxy-2-methyl-(12H)-isoquino[1,2-b]pyrrolo[3,2-f][1,3]benzoxazine-1-carboxylic acid, ethyl ester

CAS Number

23062-91-1

PubChem ID

4995951

InChI Key

VDDUJINYXKGZLV-UHFFFAOYSA-N

SMILES

CCOC(=O)C1=C(C)NC2=CC=C3OC4N(CCC5=CC(OC)=CC=C45)CC3=C12

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.

Solubility

Solvent Max Conc. mg/mL Max Conc. mM
Solubility
DMSO 39.24 100

Preparing Stock Solutions for PD 102807

The following data is based on the product molecular weight 392.45.

Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which all affect the solvent volumes required to prepare stock solutions.

Select a batch to recalculate based on the batch molecular weight:

Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 2.55 mL 12.74 mL 25.48 mL
5 mM 0.51 mL 2.55 mL 5.10 mL
10 mM 0.25 mL 1.27 mL 2.55 mL
50 mM 0.05 mL 0.25 mL 0.51 mL

Calculators

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Background References

References are publications that support the biological activity of the product. See our Citations tab to view 24 publications citing the usage of this product.

Product Documents for PD 102807

Certificate of Analysis

To download a Certificate of Analysis, please enter a lot or batch number in the search box below.

Product Specific Notices for PD 102807

For research use only

Customer Reviews for PD 102807 (1)

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  • Excellent product
    Name: Gaurang Trivedi
    Species: Mouse
    Assay Type: In Vitro
    Verified Customer | Posted 06/21/2019
    Used it to test on mice as well as stem cells

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