PD 173212

Discontinued Product

3552 has been discontinued.
View all Cav2.x Channel Blockers products.
PD 173212 | CAS No. 217171-01-2 | Cav2.x Channel Blockers
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Description: Potent CaV2.2 blocker

Chemical Name: N-[[4-(1,1-Dimethylethyl)phenyl]methyl-N-methyl-L-leucyl-N-(1,1-dimethylethyl)-O-phenylmethyl)-L-tyrosinamide

Purity: ≥98%

Product Details

Biological Activity

PD 173212 is a potent N-type voltage-gated calcium channel blocker (IC50 = 36 nM). Displays selectivity over K+, Na+ and L-type Ca2+ channels. Prevents tonic seizures in the audiogenic seizure model in vivo.

Technical Data

Soluble to 100 mM in DMSO and to 100 mM in ethanol
Store at +4°C

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.

Background References

  1. Structure-activity relationships of N-methyl-N-aralkyl-peptidylamines as novel N-type calcium channel blockers.
    Hu et al.
    Bioorg.Med.Chem.Letts., 1999;9:2151

Product Datasheets

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