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PDZ1 Domain inhibitor peptide

   
Product Datasheet
Catalog Number:2207
Chemical Name:
Product Details
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Biological Activity
Novel cyclic peptide that disrupts interaction between GluK2 (formally GluR6) and the postsynaptic density protein 95 (PSD-95). Competes with the C-terminus of GluK2 for binding to the PDZ1 domain of PSD-95. Inhibits clustering of kainate receptors.

Please refer to IUPHAR Guide to Pharmacology for the most recent naming conventions.

Technical Data
  • M.Wt:
    819.95
  • Formula:
    C38H61N9O11
  • Sequence:
    YKKTEAV

    (Modifications: Ala-6 = β-Ala, Cyclized = Lys-3 - Ala-6))

  • Solubility:
    Soluble to 1 mg/ml in 5% acetonitrile / water and to 4 mg/ml in DMSO
  • Storage:
    Desiccate at -20°C
  • CAS No:
    1315378-73-4
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis. All Tocris products are intended for laboratory research use only.
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