PDZ1 Domain inhibitor peptide

Tocris Bioscience | Catalog # 2207

Disrupts interaction between GluK2 and PSD-95 PDZ1 domain
Tocris Bioscience
Discontinued Product
2207 has been discontinued. View all Kainate Receptor Peptides products.

Key Product Details

Description

Disrupts interaction between GluK2 and PSD-95 PDZ1 domain
View all Kainate Receptor Peptides »

Product Description

PDZ1 Domain inhibitor peptide is a novel cyclic peptide that disrupts interaction between GluK2 (formerlyy GluR6) and the postsynaptic density protein 95 (PSD-95). Competes with the C-terminus of GluK2 for binding to the PDZ1 domain of PSD-95. Inhibits clustering of kainate receptors.

Please refer to IUPHAR Guide to Pharmacology for the most recent naming conventions.

Product Specifications for PDZ1 Domain inhibitor peptide

Molecular Weight

819.95

Formula

C38H61N9O11

Storage

Desiccate at -20°C

CAS Number

1315378-73-4

PubChem ID

90488746

InChI Key

XXRRADBJCXMGOW-RMLJCASOSA-N

SMILES

[H]N[C@@H](CC1=CC=C(O)C=C1)C(=O)N[C@@H](CCCCN)C(=O)N[C@H]1CCCCNC(=O)CC[C@H](NC(=O)[C@@H](NC1=O)[C@@H](C)O)C(=O)N[C@@H](C)C(=O)N[C@@H](C(C)C)C(O)=O

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.

Solubility

Solubility Soluble to 4mg/ml in DMSO and to 1mg/ml in 5% acetonitrile / water

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Background References

References are publications that support the biological activity of the product.

Product Documents for PDZ1 Domain inhibitor peptide

Certificate of Analysis

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Product Specific Notices for PDZ1 Domain inhibitor peptide

For research use only

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