Perhexiline maleate

Tocris Bioscience | Catalog # 5166

Carnitine palmitoyltransferase 1 and 2 (CPT1/2) inhibitor
Tocris Bioscience

Key Product Details

Description

Carnitine palmitoyltransferase 1 and 2 (CPT1/2) inhibitor
View all Other Transferase Inhibitors »

Product Description

Perhexiline maleate is a carnitine palmitoyltransferase 1 and 2 (CPT1/2) inhibitor. Inhibits palmitate oxidation in rat cardiomyocytes and increases cardiac efficiency in isolated rat hearts. Antianginal.

Product Specifications for Perhexiline maleate

Molecular Weight

393.56

Formula

C19H35N.C4H4O4

Storage

Store at +4°C

Purity

≥98% (HPLC)

Chemical Name

2-(2,2-Dicyclohexylethyl)piperidine maleate

CAS Number

6724-53-4

PubChem ID

5284439

InChI Key

JDZOTSLZMQDFLG-BTJKTKAUSA-N

SMILES

OC(\C=C/C(O)=O)=O.C1(CC(C3CCCCC3)C2CCCCC2)NCCCC1

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.

Solubility

Solvent Max Conc. mg/mL Max Conc. mM
Solubility
DMSO 39.36 100
Ethanol 7.87 20

Preparing Stock Solutions for Perhexiline maleate

The following data is based on the product molecular weight 393.56.

Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which all affect the solvent volumes required to prepare stock solutions.

Select a batch to recalculate based on the batch molecular weight:

Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 2.54 mL 12.70 mL 25.41 mL
5 mM 0.51 mL 2.54 mL 5.08 mL
10 mM 0.25 mL 1.27 mL 2.54 mL
50 mM 0.05 mL 0.25 mL 0.51 mL

Calculators

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Background References

References are publications that support the biological activity of the product. See our Citations tab to view 3 publications citing the usage of this product.

Product Documents for Perhexiline maleate

Certificate of Analysis

To download a Certificate of Analysis, please enter a lot or batch number in the search box below.

Product Specific Notices for Perhexiline maleate

For research use only

Citations for Perhexiline maleate

Customer Reviews for Perhexiline maleate (1)

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  • CPT1 antagonism on acute brain slices
    Name: Anonymous
    Species: Mouse
    Assay Type: Ex Vivo
    Cell Line/Tissue: acute brain slice
    Verified Customer | Posted 01/10/2018
    30 minute pre-incubation, rapid effect
    Used as a second way to block CPT1 (etomoxir was the other blocker used). Both had the same effect, confirming the involvement of CPT1 in our assay.

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