Catalog Number: 5549
Chemical Name: 6-(4-Methyl-1-piperazinyl)-11H-dibenz[b,e]azepine
Biological Activity
Potent and selective hM3Dq DREADD agonist (EC50 = 2.8 nM). Exhibits >10,000-fold selectivity for hM3Dq over hM3.
Technical Data
  • M.Wt:
    291.39
  • Formula:
    C19H21N3
  • Solubility:
    Soluble to 50 mM in DMSO and to 5 mM in water with gentle warming
  • Purity:
    >99%
  • Storage:
    Store at RT
  • CAS No:
    1977-11-3
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis. All Tocris products are intended for laboratory research use only.
Background References
  1. The first structure-activity relationship studies for designer receptors exclusively activated by designer drugs.
    Chen et al.
    ACS Chem.Neurosci., 2015;18:476

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