Discontinued Product
2024 has been discontinued.
View all mu Opioid Receptor Agonists products.
Product Description
Selective μ opioid receptor agonist (IC50 values are 5.5 and > 10000 nM for inhibition of 125I-FK 33,824 and 125I-DADLE binding to μ and δ sites respectively). Produces naloxone-reversible analgesia, catalepsy and hyperthermia following central administration in rats in vivo.
Product Specifications for PL 017
Molecular Weight
535.64
Formula
C29H37N5O5
Storage
Store at -20°C
CAS Number
83397-56-2
PubChem ID
10437173
InChI Key
JAKBYSTWCHUQOK-QORCZRPOSA-N
SMILES
[H]N[C@@H](CC1=CC=C(O)C=C1)C(=O)N1CCC[C@H]1C(=O)N(C)[C@@H](CC1=CC=CC=C1)C(=O)N1CCC[C@H]1C(N)=O
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
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Solubility
| Solubility | Soluble to 1mg/ml in water |
Calculators
Background References
References are publications that support the biological activity of the product.
- Meyer and Meyer Behavioral effects of the μ-opioid peptide agonists DAMGO, DALDA and PL017 on locomotor activities. Pharmacol.Biochem.Behav. 1993 PMID: 8265694
- Xin Body temperature and analgesic effects of selective mu and kappa opioid receptor agonists microdialyzed into rat brain. J.Pharmacol.Exp.Ther. 1997 PMID: 9103537
- Chang Potent morphiceptin analogs: structure activity relationships and morphine-like activities. J.Pharmacol.Exp.Ther. 1983 PMID: 6313901
Product Documents for PL 017
Certificate of Analysis
To download a Certificate of Analysis, please enter a lot or batch number in the search box below.
Product Specific Notices for PL 017
For research use only
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