Potent and selective adenosine A2B
receptor antagonist (IC50
= 3.64 nM at human A2B
receptors).� Displays > 100-fold selectivity over hA1
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All Tocris products are intended for laboratory research use only.
1-alkyl-8-(piperazine-1-sulfonyl)phenylxanthines: development and characterization of adenosine A2B receptor antagonists and a new radioligand with subnanomolar affinity and subtype specificity.
Borrmann et al.