Home / Histamine H3 Receptor Antagonists / ROS 234 dioxalate

ROS 234 dioxalate

2034 Datasheet / COA / SDS
Catalog # Availability Size / Price Qty
2034/10
2034/50
ROS 234 dioxalate | CAS No. 1781941-93-2 | Histamine H3 Receptor Antagonists
1 Image
Description: Potent H3 antagonist

Chemical Name: N-[3-(1H-Imidazol-4-yl)propyl]-1H-benzimidazol-2-amine dioxalate

Purity: ≥99%

Product Details
Supplemental Products
Reviews
Biological Activity Technical Data Background Product Datasheets Calculators

Biological Activity

Potent H3 antagonist (pKB at guinea-pig ileum H3-receptor = 9.46). Limited blood brain barrier permeability (ED50 = 19.12 mg/kg i.p.).

Technical Data

M.Wt:
421.37
Formula:
C13H15N5.2C2H2O4
Solubility:
Soluble to 50 mM in water and to 50 mM in DMSO
Purity:
≥99%
Storage:
Desiccate at RT
CAS No:
1781941-93-2

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.

Background References

  1. CNS access of selected H3-antagonists: ex vivo binding study in rats.
    Ballabeni et al.
    Inflamm.Res., 2002;51:S55
  2. Synthesis, biological activity, QSAR and QSPR study of 2-aminobenzimidazole derivatives as potent H3-antagonists.
    Mor et al.
    Bioorg.Med.Chem.Lett., 2004;12:663

Product Datasheets

Reconstitution Calculator
Molarity Calculator

Reconstitution Calculator

The reconstitution calculator allows you to quickly calculate the volume of a reagent to reconstitute your vial. Simply enter the mass of reagent and the target concentration and the calculator will determine the rest.

=
÷

Molarity Calculator

=
x
x
g/mol

*When preparing stock solutions always use the batch-specific molecular weight of the product found on the vial label and SDS / CoA (available online).

FAQs

No product specific FAQs exist for this product, however you may

View all Small Molecule FAQs

VersaClone cDNA Plasmids

Human Histamine H3 R (NP_009163) VersaClone cDNA

RDC0344

Mouse Histamine H3 R (NP_598610) VersaClone cDNA

RDC0728

Reviews for ROS 234 dioxalate

There are currently no reviews for this product. Be the first to review ROS 234 dioxalate and earn rewards!

Have you used ROS 234 dioxalate?

Submit a review and receive an Amazon gift card.

$25/€18/£15/$25CAN/¥75 Yuan/¥1250 Yen for a review with an image

$10/€7/£6/$10 CAD/¥70 Yuan/¥1110 Yen for a review without an image

Submit a Review
Tocris Bioscience is the leading supplier of novel and exclusive tools for life science research with over 30 years' experience in the industry. Tocris is a Bio-Techne brand.