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SAH-EZH2

Catalog #: 6708 Datasheet / COA / SDS

Discontinued Product

6708 has been discontinued.
View all EZH2 Inhibitor products.
SAH-EZH2
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Description: EZH2/EDD interaction inhibitor; suppresses PCR2 complex function
Product Details
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Biological Activity Technical Data Additional Information Background Product Datasheets Calculators

Biological Activity

SAH-EZH2 is an EZH2/EPP interaction inhibitor (Kd = 320 nM). Suppresses EZH2 expression and H3K27 trimethylation by PCR2 complex. Arrests proliferation and induces monocyte to macrophage differentiation of MLL-AF9 leukemia cell line.

Technical Data

M.Wt:
3432.05
Formula:
C155H256N48O40
Sequence:
FSSNRXKILXRTQILNQEWKQRRIQPV

(Modifications: Phe-1 = N-terminal Ac, X = (S)-2-(4-pentenyl)alanine, X-6 and X-10 stapled together with a double bond)

Solubility:
Soluble to 1 mg/ml in water
Storage:
Store at -20°C
CAS No:
1453222-26-8

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.

Additional Information

Licensing Caveats:
Sold under license from Dana-Farber Cancer Institute

Product Datasheets

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Reconstitution Calculator

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