SB 205607 dihydrobromide
Chemical Name: (R*,S*)-(±)-2-Methyl-4aa-(3-hydroxyphenyl)-1,2,3,4,4a,5,12,12aa-octahydroquinolino[2,3,3-g]isoquinoline dihydrobromide
Biological ActivityThe first described non-peptide δ1 opioid receptor agonist with very high affinity and selectivity for the δ1 subtype (Ki values are 1.12, 2320 and 1790 nM at δ1, μ and κ receptors respectively).
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Antinociceptive effects of the selective non-peptidic δ-opioid receptor agonist TAN-67 in diabetic mice.
Kamei et al.
The pharmacological profile of δ opioid receptor ligands (+) and (-) TAN-67 on pain modulation.
Nagase et al.
Life Sci., 2001;68:2227
Properties of TAN-67, a non-peptidic β-opioid receptor agonist, at cloned human δ- and μ-opioid receptors.
Knap et al.
Syntheses of non-peptidic delta opioid agonists and their structure-activity relationships.
Nagase et al.
Jpn.J.Pharmacol., 1994;64:Suppl. 1, 35P
Citations for SB 205607 dihydrobromide
The citations listed below are publications that use Tocris products. Selected citations for SB 205607 dihydrobromide include:
2 Citations: Showing 1 - 2
Critical Role for Gi/o-Protein Activity in the Dorsal Striatum in the Reduction of Voluntary Alcohol Intake in C57Bl/6 Mice.
Authors: Robins Et al.
Front Psychiatry 2018;9:112
The delta opioid receptor antagonist, SoRI-9409, decreases yohimbine stress-induced reinstatement of ethanol-seeking.
Authors: Nielsen Et al.
Addict Biol 2012;17:224
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