SB 205607 dihydrobromide

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0921/10
SB 205607 dihydrobromide | CAS No. 1217628-73-3 | delta Opioid Receptor Agonists
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Description: Selective, high affinity non-peptide δ1 agonist
Alternative Names: TAN 67

Chemical Name: (R*,S*)-(±)-2-Methyl-4aa-(3-hydroxyphenyl)-1,2,3,4,4a,5,12,12aa-octahydroquinolino[2,3,3-g]isoquinoline dihydrobromide

Purity: ≥97%

Product Details
Citations (2)
Supplemental Products
Reviews

Biological Activity

The first described non-peptide δ1 opioid receptor agonist with very high affinity and selectivity for the δ1 subtype (Ki values are 1.12, 2320 and 1790 nM at δ1, μ and κ receptors respectively).

Technical Data

M.Wt:
506.28
Formula:
C23H24N2O.2HBr
Solubility:
Soluble to 100 mM in water and to 100 mM in DMSO
Purity:
≥97%
Storage:
Store at RT
CAS No:
1217628-73-3

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.

Additional Information

Licensing Caveats:
Sold under license

Background References

  1. Antinociceptive effects of the selective non-peptidic δ-opioid receptor agonist TAN-67 in diabetic mice.
    Kamei et al.
    Eur.J.Pharmacol., 1995;276:131
  2. The pharmacological profile of δ opioid receptor ligands (+) and (-) TAN-67 on pain modulation.
    Nagase et al.
    Life Sci., 2001;68:2227
  3. Properties of TAN-67, a non-peptidic β-opioid receptor agonist, at cloned human δ- and μ-opioid receptors.
    Knap et al.
    Eur.J.Pharmacol., 1995;291:129
  4. Syntheses of non-peptidic delta opioid agonists and their structure-activity relationships.
    Nagase et al.
    Jpn.J.Pharmacol., 1994;64:Suppl. 1, 35P

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Citations for SB 205607 dihydrobromide

The citations listed below are publications that use Tocris products. Selected citations for SB 205607 dihydrobromide include:

2 Citations: Showing 1 - 2

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