Sitagliptin phosphate

Catalog # Availability Size / Price Qty
6816/50
6816/10
DPPIV/CD26 Inhibitors Small Molecule
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Description: Potent and selective DPP IV inhibitor

Chemical Name: (3R)-3-Amino-1-[5,6-dihydro-3-(trifluoromethyl)-1,2,4-triazolo[4,3-a]pyrazin-7(8H)-yl]-4-(2,4,5-trifluorophenyl)-1-butanone phosphate

Purity: ≥98%

Product Details
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Biological Activity

Potent and selective DPP IV (DPP4) inhibitor (IC50 = 18 nM). Displays >2600-fold selectivity for DDP IV over other proline specific peptidases. Reduces blood glucose and increases GLP-1 levels after oral glucose tolerance test in normal and diet-induced obese mice.

Technical Data

M.Wt:
505.31
Formula:
C16H15F6N5O.H3O4P
Solubility:
Soluble to 50 mM in water and to 50 mM in DMSO
Purity:
≥98%
Storage:
Desiccate at RT
CAS No:
654671-78-0

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.

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