TC-C 14G

Key Product Details

Product Description

TC-C 14G is a potent, high affinity CB₁ receptor inverse agonist (EC₅₀ = 11 nM in cAMP assay; K_i = 4 nM). Demonstrates high efficacy in a hypothermia assay (ID₅₀ = 5 mg/kg) in vivo.

Product Specifications for TC-C 14G

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.

Solubility

Preparing Stock Solutions for TC-C 14G

The following data is based on the product molecular weight 492.30.

Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which all affect the solvent volumes required to prepare stock solutions.

Select a batch to recalculate based on the batch molecular weight:

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Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
1 mM	2.03 mL	10.16 mL	20.31 mL
5 mM	0.41 mL	2.03 mL	4.06 mL
10 mM	0.20 mL	1.02 mL	2.03 mL
50 mM	0.04 mL	0.20 mL	0.41 mL

Calculators

Background References

References are publications that support the biological activity of the product.

• Alig Benzodioxoles: novel cannabinoid-1 receptor inverse agonists for the treatment of obesity. J.Med.Chem. 2008 PMID: 18335976

Product Documents for TC-C 14G