Blocker of Kir
1.1 channels; displays >250-fold selectivity for Kir
values are 1.1, 274 and 361 nM for Kir
3.1/3.2 and Kir
3.1/3.4 respectively). Derivative of tertiapin-Q
(Cat. No. 1316).
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
All Tocris products are intended for laboratory research use only.
Engineered specific and high-affinity inhibitor for a subtype of inward-rectifier K+ channels.
Ramu et al.