Tertiapin LQ

Tocris Bioscience | Catalog # 4339

Selective Kir1.1 blocker; derivative of tertiapin-Q (Cat. No. 1316)
Tocris Bioscience
Discontinued Product
4339 has been discontinued. View all Inward Rectifier Potassium Channel Blockers products.

Key Product Details

Description

Selective Kir1.1 blocker; derivative of tertiapin-Q (Cat. No. 1316)
View all Inward Rectifier Potassium Channel Blockers »

Product Description

Tertiapin LQ is a blocker of Kir1.1 channels; displays >250-fold selectivity for Kir1.1 (Kd values are 1.1, 274 and 361 nM for Kir1.1, Kir3.1/3.2 and Kir3.1/3.4 respectively). Derivative of tertiapin-Q (Cat. No. 1316).

Product Specifications for Tertiapin LQ

Molecular Weight

2428.03

Formula

C106H179N33O24S4

Storage

Store at -20°C

PubChem ID

90488935

InChI Key

WUMIWMIQOSXVPZ-ZPWFPUPGSA-N

SMILES

[H]N[C@@H](C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@H]1CSSC[C@@H]2NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H]3CCCN3C(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CSSC[C@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CC3=CNC4=C3C=CC=C4)NC2=O)C(=O)NCC(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(N)=O)NC(=O)[C@H](CC(N)=O)NC1=O)[C@@H](C)CC)[C@@H](C)CC)[C@@H](C)CC

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.

Solubility

Solubility Soluble to 2mg/ml in 20% acetonitrile / water

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Background References

References are publications that support the biological activity of the product.

Product Documents for Tertiapin LQ

Certificate of Analysis

To download a Certificate of Analysis, please enter a lot or batch number in the search box below.

Product Specific Notices for Tertiapin LQ

For research use only

Related Research Areas

Ion Channels and Regulators

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