UFP-101

  ( 2 citations )    
Product Datasheet
Catalog Number:1552
Alternate Names:[Nphe1,Arg14,Lys15]Nociceptin-NH2
Chemical Name:
Product Details
Citations (2)
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Biological Activity
Potent, selective and competitive silent antagonist for the NOP opioid receptor. Binds to NOP with high affinity (pKi = 10.24) and displays > 3000-fold selectivity over δ, μ and κ opioid receptors. Antinociceptive and opposes the action of nociceptin in vivo.
Technical Data
  • M.Wt:
    1908.19
  • Formula:
    C82H138N32O21
  • Sequence:
    GGGFTGARKSARKRKNQ

    (Modifications: Gly-1 = N-(Bn)Gly, Gln-17 = C-terminal amide)

  • Solubility:
    Soluble to 1 mg/ml in water
  • Storage:
    Desiccate at -20°C
  • CAS No:
    849024-68-6
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis. All Tocris products are intended for laboratory research use only.
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Citations:

The citations listed below are publications that use Tocris products. Selected citations for UFP-101 include:

2 Citations: Showing 1 - 2
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  1. Modulation of silent and constitutively active nociceptin/orphanin FQ receptors by potent receptor antagonists and Na+ ions in rat sympathetic neurons.
    Authors: Mahmoud Et al.
    Mol Pharmacol  2010;77:804
  2. Evidence in locomotion test for the functional heterogeneity of ORL-1 receptors.
    Authors: Kuzmin Et al.
    Br J Pharmacol  2004;141:132

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VersaClone cDNA Plasmids
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Human ORL1/OPRL1 (NP_000904) VersaClone cDNA

RDC0163
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