VU 6001966

Catalog # Availability Size / Price Qty
6928/5
VU 6001966 | CAS No. 2009052-76-8 | Group II mGluR Modulators
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Description: Potent and selective negative allosteric modulator of mGlu2 receptors

Purity: ≥98%

Product Details
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Biological Activity

VU 6001966 is a potent and selective mGlu2 negative allosteric modulator (IC50 = 78 nM). Exhibits > 350-fold selectivity for mGlu2 over mGlu3. Also exhibits selectivity over other mGluRs and a panel of GPCRs, ion channels and transporters. CNS penetrant.

Technical Data

M.Wt:
326.33
Formula:
C17H15FN4O2
Solubility:
Soluble to 100 mM in DMSO and to 5 mM in ethanol
Purity:
≥98%
Storage:
Store at -20°C
CAS No:
2009052-76-8

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.

Additional Information

Licensing Caveats:
Sold under license from Vanderbilt University

Product Datasheets

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