Potent histamine H3
receptor silent antagonist (pKi
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All Tocris products are intended for laboratory research use only.
Identification of 4-(1H-imidazol-4(5)-ylmethyl)pyridine (immethridine) as a novel, potent, and highly selective histamine H3 receptor agonist.
Kitbunnadaj et al.
The histamine H3 receptor: from gene cloning to H3 receptor drugs.
Leurs et al.
Nat.Rev.Drug Discov., 2005;4:107
Constitutive activity of H3 autoreceptors modulates histamine synthesis in rat brain through the cAMP/PKA pathway.
Moreno-Delgado et al.