WEB 2086

Catalog # Availability Size / Price Qty
2339/10
2339/1
WEB 2086 | CAS No. 105219-56-5 | Platelet-activating Factor Receptor Antagonists
1 Image
Description: Potent PAF receptor antagonist
Alternative Names: Apafant

Chemical Name: 4-[3-[4[(2-Chlorophenyl)-9-methyl-6H-thieno[3,2-f][1,2,4]triazolo[4,3-a]diazepin-2-yl]-1-oxopropyl]morpholine

Purity: ≥99%

Product Details
Citations (6)
Supplemental Products
Reviews

Biological Activity

Potent, selective platelet-activating factor (PAF) receptor antagonist (Ki = 16.3 nM). Displays anti-inflammatory, antiangiogenic and anticancer activity. Inhibits growth and proliferation of MCF-7 breast cancer cells.

Technical Data

M.Wt:
455.96
Formula:
C22H22N5O2SCl
Solubility:
Soluble to 100 mM in DMSO and to 100 mM in ethanol with gentle warming
Purity:
≥99%
Storage:
Desiccate at +4°C
CAS No:
105219-56-5

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.

Product Datasheets

or select another batch:
Reconstitution Calculator
Molarity Calculator

Reconstitution Calculator

The reconstitution calculator allows you to quickly calculate the volume of a reagent to reconstitute your vial. Simply enter the mass of reagent and the target concentration and the calculator will determine the rest.

=
÷

Molarity Calculator

=
x
x
g/mol

*When preparing stock solutions always use the batch-specific molecular weight of the product found on the vial label and SDS / CoA (available online).

FAQs

No product specific FAQs exist for this product, however you may

View all Small Molecule FAQs

Reviews for WEB 2086

There are currently no reviews for this product. Be the first to review WEB 2086 and earn rewards!

Have you used WEB 2086?

Submit a review and receive an Amazon gift card.

$25/€18/£15/$25CAN/¥75 Yuan/¥1250 Yen for a review with an image

$10/€7/£6/$10 CAD/¥70 Yuan/¥1110 Yen for a review without an image

Submit a Review
Tocris Bioscience is the leading supplier of novel and exclusive tools for life science research with over 30 years' experience in the industry. Tocris is a Bio-Techne brand.