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1 result for "mAChR M2 Receptor Modulators Small Molecules and Peptides" in Products
mAChR M2 Receptor Modulators Small Molecules and Peptides
M2 receptors are members of the G-protein-coupled receptor (GPCR) family which are found mostly bound to Gi proteins, generally leading to inhibitory effects. They are one of five muscarinic receptors that act to control the metabotropic functions of acetylcholine (ACh) in the central nervous system (CNS). M2 receptors are densely populated in the heart, airway smooth muscle, the hippocampus and most other brain regions.
Activation of the M2 receptor leads to several responses, including the ...
Positive allosteric modulator of M2 and M4 receptors
| Chemical Name: | 3-Amino-5-chloro-N-cyclopropyl-4-methyl-6-[2-(4-methyl-1-piperazinyl)-2-oxoethoxy]-thieno[2,3-b]pyridine-2-carboxamide |
| Purity: | ≥98% |
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