2 results for "NTS2/NTSR2" in Products

NTS2/NTSR2 Products

Binding and pharmacological studies demonstrate that NTSR2 binds neurotensin as well as several other ligands already described for NTSR1. Unlike NTSR1, NTSR2 recognizes, with high affinity, levocabastine, a histamine H1 receptor antagonist previously shown to compete with neurotensin for low-affinity binding sites in brain. NTSR2 may be of physiological importance and a natural agonist for the receptor may exist.

Highly potent NTS receptor antagonist

Chemical Name: 2-[[[5-(2,6-Dimethoxyphenyl)-1-[4-[[[3-(dimethylamino)propyl]methylamino]carbonyl]-2-(1-methylethyl)phenyl]-1H-pyrazol-3-yl]carbonyl]amino]-tricyclo[3.3.1.13,7]decane-2-carboxylic acid
Purity: ≥97%
Highly potent NTS receptor antagonist
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Potent and selective non-peptide NTS2 antagonist

Chemical Name: N-[2-[5-[[(4-Methylphenyl)sulfonyl]amino]-3-(2,2,2-trifluoroacetyl)-1H-indol-1-yl]acetyl]-L-leucine
Purity: ≥98%
Potent and selective non-peptide NTS2 antagonist
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