Potent non-peptide neurotensin (NT) receptor antagonist that binds with high affinity (IC50
= 0.32 - 3.96 nM; Ki
< 10 nM). Attenuates amphetamine-induced hyperactivity and is orally active in vivo
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All Tocris products are intended for laboratory research use only.
Biochemical and pharmacological activities of SR 142948A, a new potent neurotensin receptor antagonist.
Gully et al.
X-ray structural characterization of SR 142948, a novel potent synthetic neurotensin receptor antagonist.
Quere et al.
Effects of the selective neurotensin antagonist SR 142948A on 3,4-methylenedioxymethamphetamine-induced behaviours in mice.
Marie-Claire et al.
The citations listed below are publications that use Tocris products. Selected citations for SR 142948 include:
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