5 results for "additional-p53-related-compounds&view=expanded" in 产品

Restores mutant p53 activity; proapoptotic

Chemical Name: 1-[(1-Oxopropoxy)methyl]-1H-pyrrole-2,5-dione
Restores mutant p53 activity; proapoptotic
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Restores mutant p53 activity

Alternate Names: APR-246
Chemical Name: 2-(Hydroxymethyl)-2-(methoxymethyl)-1-azabicyclo[2.2.2]octan-3-one
Purity: ≥98%
Restores mutant p53 activity
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p53 inhibitor. Also aryl hydrocarbon receptor agonist

Chemical Name: 1-(4-Methylphenyl)-2-(4,5,6,7-tetrahydro-2-imino-3(2H)-benzothiazolyl)ethanone hydrobromide
p53 inhibitor. Also aryl hydrocarbon receptor agonist
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Selective exportin-1 (XPO1/CRM1) inhibitor

Chemical Name: (2Z)-3-[3-[3,5-Bis(trifluoromethyl)phenyl]-1H-1,2,4-triazol-1-yl]-2-propenoic acid 2-(2-pyridinyl)hydrazide
Purity: ≥98%
Selective exportin-1 (XPO1/CRM1) inhibitor
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RNA polymerase I inhibitor; also p53 pathway activator

Chemical Name: N-[2-(Dimethylamino)ethyl]-12-oxo-12H-benzo[g]pyrido[2,1-b]quinazoline-4-carboxamide
Purity: ≥98%
RNA polymerase I inhibitor; also p53 pathway activator
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