26 results for "GABA A R alpha 3" in 产品

GABA A R alpha 3 Products

Gamma-aminobutyric acid (GABA) is the primary inhibitory neurotransmitter in the central nervous system, causing a hyperpolarization of the membrane through the opening of a Cl- channel associated with the GABAA receptor (GABAA-R) subtype. GABAA-Rs are important therapeutic targets for a range of sedative, anxiolytic, and hypnotic agents and are implicated in several diseases including epilepsy, anxiety, depression, and sub-stance abuse. The GABAA-R is a multimeric subunit complex. To date six ...

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Reactivity: Human
Applications:
R&D Systems VersaClone cDNA Plasmids
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Reactivity: Human, Mouse
Details: Rabbit IgG Polyclonal
Applications: IHC, WB
Western Blot: GABA-AR alpha 3 Antibody [NBP1-87499]
(9)
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Reactivity: Mouse, Rat
Details: Rabbit IgG Polyclonal
Applications: KO, IHC, WB, ICC/IF
Western Blot: GABA-AR alpha 3 Antibody [NB100-61096]
(2)
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Reactivity: Human
Applications:
R&D Systems VersaClone cDNA Plasmids
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Reactivity: Human
Applications:
R&D Systems VersaClone cDNA Plasmids
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Reactivity: Human, Mouse, Rat
Details: Rabbit IgG Polyclonal
Applications: WB
Western Blot: GABA-AR alpha 3 AntibodyAzide and BSA Free [NBP3-03646]
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Reactivity: Human, Mouse, Rat
Details: Rabbit IgG Polyclonal
Applications: WB, ELISA
GABA-AR alpha 3 Antibody - BSA Free
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Reactivity: Human
Source: Wheat germ
Applications: WB, ELISA, AP, MA
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Reactivity: Human
Source: Wheat germ
Applications: WB, ELISA, AP, MA
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Reactivity: Human
Details: Rabbit Polyclonal
Applications: IHC
Immunohistochemistry-Paraffin: GABA-AR alpha 3 Antibody [NBP3-14326]
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Reactivity: Human
Details: Rabbit Polyclonal
Applications: IHC
Immunohistochemistry-Paraffin: GABA-AR alpha 3 Antibody [NBP3-14327]
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Reactivity: Human
Applications: WB
Western Blot: GABA-AR alpha 3 Overexpression Lysate [NBL1-10916]
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Reactivity: Human
Source: E. coli
Applications: AC
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Competitive and selective GABAA antagonist

Alternate Names: Gabazine
Chemical Name: 6-Imino-3-(4-methoxyphenyl)-1(6H)-pyridazinebutanoic acid hydrobromide
Purity: ≥98%
Competitive and selective GABAA antagonist
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Potent GABAA agonist; also GABAA-ρ partial agonist

Chemical Name: 5-Aminomethyl-3-hydroxyisoxazole
Purity: ≥98%
Potent GABAA agonist; also GABAA-ρ partial agonist
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GABAA agonist

Alternate Names: Gaboxadol
Chemical Name: 4,5,6,7-Tetrahydroisoxazolo[5,4-c]pyridin-3-ol hydrochloride
Purity: ≥98%
GABAA agonist
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Benzodiazepine inverse agonist

Chemical Name: N-Methyl-β-carboline-3-carboxamide
Purity: ≥99%
Benzodiazepine inverse agonist
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Benzodiazepine antagonist

Alternate Names: Ro 15-1788
Chemical Name: 8-Fluoro-5,6-dihydro-5-methyl-6-oxo-4H-imidazo[1,5-a][1,4]benzodiazepine-3-carboxylic acid, ethyl ester
Purity: ≥99%
Benzodiazepine antagonist
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α5-selective GABAA inverse agonist

Chemical Name: 3-(1,1-Dimethylethyl)-7-(5-methyl-3-isoxazolyl)-2-[(1-methyl-1H-1,2,4-triazol-5-yl)methoxy]-pyrazolo[1,5-d][1,2,4]triazine
Purity: ≥98%
α5-selective GABAA inverse agonist
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GABAA partial agonist; displays subtype selectivity

Chemical Name: 3-(2,5-Difluorophenyl)-7-(1,1-dimethylethyl)-6-[(1-methyl-1H-1,2,4-triazol-5-yl)methoxy]-1,2,4-triazolo[4,3-b]pyridazine
Purity: ≥98%
GABAA partial agonist; displays subtype selectivity
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Postitive allosteric modulator of GABAA receptors

Chemical Name: (3α,5β)-3-Hydroxy-pregnan-20-one
Postitive allosteric modulator of GABAA receptors
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Positive allosteric modulator of GABAA receptors

Alternate Names: 3a,5a-THPROG
Chemical Name: (3α,5α)-3-Hydroxy-pregnan-20-one
Positive allosteric modulator of GABAA receptors
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Active metabolite of oxcarbazepine (Cat. No. 3864)

Alternate Names: GP 47779
Chemical Name: 10,11-Dihydro-10-hydroxy-5H-dibenz(Z)[b,f]azepin-5-carboxamide
Purity: ≥98%
Active metabolite of oxcarbazepine (Cat. No. 3864)
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Benzodiazepine inverse agonist

Chemical Name: 4-Ethyl-6,7-dimethoxy-9H-pyrido[3,4-b]indole-3-carboxylic acid methyl ester hydrochloride
Purity: ≥98%
Benzodiazepine inverse agonist
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Benzodiazepine partial inverse agonist

Chemical Name: 8-Azido-5,6-dihydro-5-methyl-6-oxo-4H-imidazo[1,5-a][1,4]benzodiazepine-3-carboxylic acid ethyl ester
Purity: ≥98%
Benzodiazepine partial inverse agonist
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