4 results for "Sigma1 Receptor Ligands Small Molecules and Peptides" in 产品

Sigma1 Receptor Ligands Small Molecules and Peptides

σ1 receptors are members of the σ family of receptors that also includes σ2 receptors. Originally thought to be opioid receptors or the phencyclidine binding site on the NMDA receptor, they are now known to be distinct targets. These receptors are distinguished from σ2 receptors as they exhibit high affinity and stereoselectivity for the (+)-isomers of pentazocine, SK&F 10047 and cyclazocine, as well as having different tissue distribution patterns and subcellular ...

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Dopamine antagonist; displays some D2 selectivity

Chemical Name: 4-[4-(4-Chlorophenyl)-4-hydroxy-1-piperidinyl]-1-(4-fluorophenyl)-1-butanone hydrochloride
Purity: ≥98%
Dopamine antagonist; displays some D2 selectivity
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Selective σ1 ligand, putative antagonist

Chemical Name: 1-[2-(3,4-Dichlorophenyl)ethyl]-4-methylpiperazine dihydrochloride
Purity: ≥99%
Selective σ1 ligand, putative antagonist
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5-HT reuptake inhibitor

Chemical Name: (E)-5-Methoxy-1-[4-(trifluoromethyl)phenyl]-1-pentanone-O-(2-aminoethyl)oxime maleate
Purity: ≥99%
5-HT reuptake inhibitor
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Selective σ1 ligand; antidepressant

Chemical Name: (R)-(+)-N-Cyclopropylmethyl-α-ethyl-N-methyl-α-[(2E)-3-phenyl-2-propenyl)benzenemethanamine hydrochloride
Purity: ≥98%
Selective σ1 ligand; antidepressant
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