Potent, high affinity H4
receptor agonist (Ki
= 7 nM) that displays > 100-fold selectivity over other human histamine receptor subtypes.
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
All Tocris products are intended for laboratory research use only.
Evaluation of histamine H1-, H2-, and H3-receptor ligands at the human histamine H4 receptor: identification of 4-methylhistamine as the first potent and selective H4 receptor agonist.
Lim et al.
Compared pharmacology of human histamine H3 and H4 receptors: structure-activity relationships of histamine derivatives.
Gbahou et al.
The citations listed below are publications that use Tocris products. Selected citations for 4-Methylhistamine dihydrochloride include:
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