Biological Activity High affinity and selective CB1 antagonist (Kd = 0.89 nM). Exhibits 100-fold selectivity for CB1 over CB2. Attenuates CB1 agonist AM 411-induced locomotor suppression and reduces food intake in vivo, but does not induce signs of nausea.
Soluble to 20 mM in DMSO and to 20 mM in ethanol
Store at +4°C
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