B-HT 933 dihydrochloride

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B-HT 933 dihydrochloride | CAS No. 36067-72-8 | Adrenergic alpha-2 Receptor Agonists
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Description: Selective α2 agonist
Alternative Names: Azepexole

Chemical Name: 6-Ethyl-5,6,7,8-tetrahydro-4H-oxazolo[4,5-d]azepin-2-amine dihydrochloride

Purity: ≥99%

Product Details
Citations (1)
Supplemental Products

Biological Activity

B-HT 933 dihydrochloride is a selective α2-adrenoceptor agonist. Exhibits greater than 300-fold selectivity for the α2-adrenoceptor over the α1-adrenoceptor.

Technical Data

Soluble to 100 mM in water and to 50 mM in DMSO
Desiccate at RT

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.

Background References

  1. The thermogenic actions of α2-adrenoceptor agonists in reserpinized mice are mediated via a central postsynaptic α2-adrenoceptor mechanism.
    Bill et al.
    Br.J.Pharmacol., 1989;96:133
  2. The mechanism of action of α2-adrenoceptors in human isolated subcutaneous resistance arteries.
    Parkinson and Hughes
    Br.J.Pharmacol., 1995;115:1463
  3. Pharmacological characterization of B-HT 933 (2-amino-6-ethyl-4,5,7,8-tetrahydro-6H-oxazolo-[5,4-d]-azepindihydrochloride) as a hypotensive agent of the "clonidine-type".
    Kobinger and Pichler
    Naunyn-Schmied.Arch.Pharmacol., 1977;300:39

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Citation for B-HT 933 dihydrochloride

The citations listed below are publications that use Tocris products. Selected citations for B-HT 933 dihydrochloride include:

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