CP 376395 hydrochloride

Catalog # Availability Size / Price Qty
3212/10
3212/50
CP 376395 hydrochloride | CAS No. 1013933-37-3 | CRF1 Receptor Antagonists
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Description: Potent and selective CRF1 antagonist; binds at an allosteric site

Chemical Name: N-(1-Ethylpropyl)-3,6-dimethyl-2-(2,4,6-trimethylphenoxy)-4-pyridinamine hydrochloride

Purity: ≥99%

Product Details
Citations (3)
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Biological Activity

Potent and selective CRF1 receptor antagonist (Ki values are 12 and >10000 nM for CRF1 and CRF2 receptors respectively). Binds at an allosteric site. Attenuates CRF-induced activation of the HPA axis in vivo following i.v. administration. Orally active.

Technical Data

M.Wt:
362.94
Formula:
C21H30N2O.HCl
Solubility:
Soluble to 50 mM in water and to 100 mM in DMSO
Purity:
≥99%
Storage:
Desiccate at RT
CAS No:
1013933-37-3

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.

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Citations for CP 376395 hydrochloride

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