AMPAkine; positive allosteric modulator of AMPA. Prototypical benzamide which occupies subsite A only. Modulates channel deactivation and desensitization.
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Functional analysis of a novel positive allosteric modulator of AMPA receptors derived from a structure-based drug design strategy.
Harms et al.
Structural and functional analysis of two new positive allosteric modulators of GluA2 desensitization and deactivation.
Timm et al.
Stable expression of recombinant AMPA receptor subunits: binding affinities and effects of allosteric modulators.
Hennegriff et al.