Catalog Number: 5418
Chemical Name: 1-[2-[2,5-Dimethyl-1-(phenylmethyl)-1H-pyrrol-3-yl]-2-oxoethyl]-1,6-dihydro-6-oxo-3-pyridinecarbonitrile
Biological Activity
Selective S1P2 allosteric agonist (EC50 = 0.48 μM). Selective for S1P2 receptors over a panel of 29 other receptors and transporters.
Technical Data
  • M.Wt:
    345.39
  • Formula:
    C21H19N3O2
  • Solubility:
    Soluble to 100 mM in DMSO
  • Purity:
    >99%
  • Storage:
    Store at +4°C
  • CAS No:
    1449747-00-5
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis. All Tocris products are intended for laboratory research use only.
Background References
  1. A sphingosine 1-phosphate receptor 2 selective allosteric agonist.
    Satsu et al.
    Bioorg.Med.Chem., 2013;21:5373

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