Ec2la

Catalog # Availability Size / Price Qty
6832/10
6832/50
Ec2la | CAS No. 2244579-87-9 | Cannabinoid R2/CB2 Receptor Ligands
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Description: Positive allosteric modulator of CB2 receptors; active in vivo

Chemical Name: N-[5-Bromo-1-[(4-fluorophenyl)methyl]-1,2-dihydro-4-methyl-2-oxo-3-pyridinyl]cycloheptanecarboxamide

Purity: ≥98%

Product Details
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Biological Activity

CB2 receptor positive allosteric modulator. Enhances CP 55940 (Cat. No. 0949) and 2-Arachidonylglycerol (Cat. No. 1298)-stimulated binding of [35S]GTPγS to CB2 receptors, but has no effect in the absence of agonist. Exhibits antinociceptive effects in an animal model of neuropathic pain.

Technical Data

M.Wt:
435.33
Formula:
C21H24BrFN2O2
Solubility:
Soluble to 20 mM in DMSO
Purity:
≥98%
Storage:
Store at -20°C
CAS No:
2244579-87-9

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.

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