Reversible and non-competitive CBP/p300 inhibitor (IC50
values are 1.1 and 2.9 μ
M, respectively). Cell permeable.
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All Tocris products are intended for laboratory research use only.
A novel cell-permeable, selective, and noncompetitive inhibitor of KAT3 histone acetyltransferases from a combined molecular pruning/classical isosterism approach.
Milite et al.