21 results for "histone-acetyltransferase-inhibitors" in Products

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iP300v

Catalog #: 7584
Product Documents

Negative control for iP300w (Cat. No. 7270)

Chemical Name: (1'R,3'S)-3'-Fluoro-N-[(4-fluorophenyl)methyl]-2',3'-dihydro-5'-[1-[2-(methylamino)-2-oxoethyl]-1H-pyrazol-4-yl]-2,5-dioxo-N-[(1S)-2,2,2-trifluoro-1-methylethyl]spiro[imidazolidine-4,1'-[1H]indene]-1-acetamide
Purity: ≥98%
Negative control for iP300w (Cat. No. 7270)

NU 9056

Catalog #: 4903
(1)
Citations (38)
Product Documents

Inhibitor of KAT5 (Tip60)

Chemical Name: 5-(1,2-Thiazol-5-yldisulfanyl)-1,2-thiazole
Inhibitor of KAT5 (Tip60)

A 485

Catalog #: 6387
Citations (67)
Product Documents

Potent and selective p300/CBP inhibitor; orally bioavailable

Chemical Name: (1R)-N-[(4-Fluorophenyl)methyl]-2,3-dihydro-5-[[(methylamino)carbonyl]amino]-2',4'-dioxo-N-[(1S)-2,2,2-trifluoro-1-methylethyl]spiro[1H-indene-1,5'-oxazolidine]-3'-acetamide
Purity: ≥98%
Potent and selective p300/CBP inhibitor; orally bioavailable

MC 1

Catalog #: 8843
Product Documents

Selective EP300 Degrader (PROTAC®)

Chemical Name: (2S,4R)-1-((S)-2-(8-(2-(4-(6-((R)-2-(((S)-2-(4-Cyanophenyl)propyl)amino)-2-phenylacetamido)pyridin-3-yl)-1H-pyrazol-1-yl)acetamido)octanamido)-3,3-dimethylbutanoyl)-4-hydroxy-N-((S)-1-(4-(4-methylthiazol-5-yl)phenyl)ethyl)pyrrolidine-2-carboxamide
Purity: ≥95%
Selective EP300 Degrader (PROTAC®)

iP300w

Catalog #: 7270
Citations (4)
Product Documents

Potent p300/CBP inhibitor

Chemical Name: (1'S,3'R)-3'-Fluoro-N-[(4-fluorophenyl)methyl]-2',3'-dihydro-5'-[1-[2-(methylamino)-2-oxoethyl]-1H-pyrazol-4-yl]-2,5-dioxo-N-[(1S)-2,2,2-trifluoro-1-methylethyl]spiro[imidazolidine-4,1'-[1H]indene]-1-acetamide
Purity: ≥98%
Potent p300/CBP inhibitor

EML 425

Catalog #: 5646
Citations (2)
Product Documents

Reversible and non-competitive CBP/p300 inhibitor

Chemical Name: 5-[(4-Hydroxy-2,6-dimethylphenyl)methylene]-1,3-bis(phenylmethyl)-2,4,6(1H,3H,5H)-pyrimidinetrione
Purity: ≥98%
Reversible and non-competitive CBP/p300 inhibitor

WM 1119

Catalog #: 6692
Citations (5)
Product Documents

High affinity KAT6A (MOZ) competitive inhibitor

Chemical Name: 2-Fluoro-N'-(3-fluoro-5-(pyridin-2-yl)benzoyl)benzenesulfonohydrazide
Purity: ≥98%
High affinity KAT6A (MOZ) competitive inhibitor

WM 8014

Catalog #: 6693
Citations (1)
Product Documents

Potent and selective KAT6A and KAT6B inhibitor

Chemical Name: N'-(4-Fluoro-5-methyl-[1,1'-biphenyl]-3-carbonyl)benzenesulfonohydrazide
Purity: ≥98%
Potent and selective KAT6A and KAT6B inhibitor

WM 3835

Catalog #: 7366
(1)
Citations (3)
Product Documents

Lysine acetyltransferase HBO1 (KAT7) inhibitor

Chemical Name: N'-(4-Fluoro-5-methyl-[1,1'-biphenyl]-3-carbonyl)-3-hydroxybenzenesulfonohydrazide
Purity: ≥98%
Lysine acetyltransferase HBO1 (KAT7) inhibitor

JQAD1

Catalog #: 7682
Citations (2)
Product Documents

Potent and selective EP300 Degrader (PROTAC®)

Chemical Name: 12-((2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindolin-5-yl)amino)-N-((R)-3'-(2-((4-fluorobenzyl)((S)-1,1,1-trifluoropropan-2-yl)amino)-2-oxoethyl)-2',4'-dioxo-2,3-dihydrospiro[indene-1,5'-oxazolidin]-5-yl)dodecanamide
Purity: ≥98%
Potent and selective EP300 Degrader
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