ERGi-USU

Catalog # Availability Size / Price Qty
6632/50
Cat.No. 6632 - ERGi-USU | C13H9N3OS | CAS No. 1147-56-4
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Description: Rio2 kinase (RIOK2) inhibitor; inhibits ERG protein

Chemical Name: 1-[2-(2-Thiazolyl)diazenyl]-2-naphthalenol

Product Details
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Biological Activity

High affinity Rio Kinase 2 (RIOK2) inhibitor (Kd = 200 nM). Exhibits >6-fold selectivity for RIOK2 over a panel of 456 kinases. Inhibits ERG protein and potently inhibits growth of ERG-positive VCaP prostate cancer cells in vitro (IC50 = 169 nM) but not ERG-negative cell lines. Also inhibits growth of VCaP xenografts in mice.

Technical Data

Formula:
C13H9N3OS
Solubility:
Soluble to 100 mM in DMSO
Storage:
Store the unopened product at 2 - 8 °C. Do not use past expiration date.
CAS No:
1147-56-4

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis. All Tocris products are intended for laboratory research use only.

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