Highly potent and selective κ
-opioid agonist (IC50
= 0.04 nM) that may be selective for the putative κ2
receptor. Anti-nociceptive and neuroprotective in vivo
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Neuroprotective actions of GR89696, a highly potent and selective κ-opioid receptor agonist.
Birch et al.
GR89,696: a potent κ-opioid agonist with subtype selectivity in rhesus monkeys.
Butelman et al.
A potent new class of κ-receptor agonist: 4-substituted 1-(arylacetyl)-2-[(dialkylamino)methyl]piperazines.
Naylor et al.